Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04357
Ion Channel
Sodium channel type 3 subunit alpha
Peptide Function
Inhibitor
Gene Name
SCN3A
Activity Data (nM)
IC50
8.79 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
85.23% inhibition at 100 μM
Sequence Information
Peptide Sequence
MKGMILFISCLLLIDIVVGGKEGYLMDHEGCKLSCFIRPSGYCGRECTLKKGSSGYCAWPACYCYGLPNWVKVWDRattusnorvegicustusnorvegicusNKCGKK
Peptide UniProt Accession
Not available
UniParc
Not available
Peptide Synonyms/Alias
Tst1
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
Intracellular solution:pH 7.3/Extracellular solution:pH 7.4
Holding Potential (mV)
−120 mV
Temperature
24 °C
Test Method
Patch-clamping
Test Species
HEK293 cell (Homo sapiens embryonic kidney 293 cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available